A2AR-agonist-1

SKU: orb1710514

Description

A2AR-agonist-1 is a dual agonist of the adenosine A2A receptor and equilibrative nucleoside transporter 1 (ENT1), exhibiting high affinity with Ki values of 4.39 nM and 3.47 nM, respectively. This small molecule is utilized in research exploring neuroprotective mechanisms, including in vitro receptor binding assays and in vivo models of neurological disorders.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 41552-95-8
• MW: 410.43
• Purity: 99.82% (May vary between batches)
• Formula: C₂₀H₂₂N₆O₄
• SMILES: OC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(NCCc3c[nH]c4ccccc34)ncnc12
• Target: Adenosine Receptor
• Solubility: DMSO:90 mg/mL (219.28 mM);10% DMSO+40% PEG300+5% Tween 80+45% Saline:3.3 mg/mL (8.04 mM)

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

N-(2-(1H-Indol-3-yl)ethyl)adenosine, AdenosineReceptor, Adenosine Receptor, A2AR-agonist-1

Compound Identifiers

PubChem CID

219015