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β2AR/M-receptor agonist-2

SKU: orb1745044

Description

This dual-action MABA compound functions as a potent β2 adrenoceptor agonist (EC50=3.7 nM) and a muscarinic M3 receptor antagonist (Ki=0.73 nM). It serves as a valuable research tool for investigating bronchodilation mechanisms and potential therapeutic strategies for obstructive lung diseases like COPD in both cellular and animal models.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number1017857-38-3
MW717.31
FormulaC36H49ClN4O7S
SMILESN(C(OC1CCN(CCCCCCCCCNC[C@H](O)C2=CC(NS(C)(=O)=O)=C(O)C=C2)CC1)=O)C3=C(C=CC=C3)C4=CC(Cl)=C(O)C=C4
TargetAChR,Others,Adrenergic Receptor

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Quality Guarantee

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Key Properties

No computed properties available.

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Protocol Information

β2AR/M-receptor agonist-2 (orb1745044)

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25 mg
$ 5,140.00
50 mg
$ 6,720.00
100 mg
$ 9,030.00
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