Tertiapin

SKU: orb2645948

Description

Tertiapin is a synthetic, disulfide-stabilized bee venom peptide that potently inhibits inward-rectifying (Kir) and large-conductance calcium-activated (BK) potassium channels. It is a valuable research tool for studying channel function in vitro and in vivo, with applications in neurobiological, cardiovascular, and autoimmune disease research such as multiple sclerosis.

Research Area

Pharmacology & Drug Discovery

Key Properties

• Target: Potassium Channel
• CAS Number: 58694-52-3
• MW: 2459.1
• Formula: C₁₀₆H₁₈₀N₃₄O₂₃S₅
• SMILES: C([C@@H](C(N[C@H](C(N[C@H](C(N[C@H](C(NCC(N[C@H](C(N[C@@H](CCCCN)C(N)=O)=O)CCCCN)=O)=O)CS)=O)CCCCN)=O)CCCCN)=O)NC([C@@H](NC([C@@H](NC([C@@H](NC(=O)[C@H]1N(C([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@H](C)N)=O)CC(C)C)=O)CS)=O)CC(N)=O)=O)CS)=O)CC(N)=O)=O)CCCNC(=N)N)=O)[C@H](CC)C)=O)[C@H](CC)C)=O)[C@H](CC)C)=O)CCC1)CC2=CN=CN2)=O)CCSC)=O)CS)=O)C=3C=4C(NC3)=CC=CC4

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

16135957