Tertiapin-Q acetate

SKU: orb2308667

Description

Tertiapin-Q acetate is a synthetic derivative of the bee venom peptide tertiapin, functioning as a potent and selective blocker of BK-type calcium-activated potassium channels. This inhibitor is a valuable research tool for studying channel physiology and K+ efflux mechanisms in both cellular and animal models of neuronal, cardiovascular, and smooth muscle function.

Research Area

Pharmacology & Drug Discovery

Key Properties

• Target: Potassium Channel
• Molecular Weight: 2512.06
• Purity: 96.44%
• Formula: C₁₀₈H₁₇₉N₃₅O₂₆S₄
• SMILES: O=C([C@@]1([H])NC([C@@H](NC([C@@H](NC([C@@]2([H])N(CCC2)C([C@](NC([C@](NC([C@](NC([C@@H](NC([C@@H](NC([C@@](CSSC[C@H](NC([C@@H](NC([C@@H](NC3=O)CCCCN)=O)CCCCN)=O)C(NCC(N[C@@H](CCCCN)C(N[C@H](C(N)=O)CCCCN)=O)=O)=O)([H])NC([C@@H](NC([C@H](CSSC1)NC([C@H](CC(C)C)NC([C@@H](N)C)=O)=O)=O)CC(N)=O)=O)=O)CC(N)=O)=O)CCCNC(N)=N)=O)([H])[C@@H](C)CC)=O)([H])[C@@H](C)CC)=O)([H])[C@@H](C)CC)=O)=O)CC4=CN=CN4)=O)CCC(N)=O)=O)N[C@H]3CC5=CNC6=CC=CC=C56.CC(O)=O

Storage & Handling

• Storage: keep away from direct sunlight,keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

Tertiapin-Q acetate(910044-56-3 Free base), TertiapinQacetate(910044563Freebase), Potassium Channel, PotassiumChannel

Compound Identifiers

PubChem CID

176418977