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Pimelic Diphenylamide 106

SKU: orb1223589

Description

A slow, tight-binding inhibitor of class I HDACs (HDAC1/2/3, Ki=148/102/14 nM respectively); shows weak inhibition on HDAC8 (IC50=5 uM); has preference toward HDAC3.

Images & Validation

Key Properties

CAS Number937039-45-7
MW339.4314
Purity>98% (HPLC)
FormulaC20H25N3O2
SMILESO=C(NC1=CC=CC=C1N)CCCCCC(NC2=CC=C(C)C=C2)=O
TargetHDAC
SolubilityDMSO: ≥ 25 mg/mL

Storage & Handling

StorageStorage temperature: -20°C. Stability: ≥ 2 years
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

RGFA-8 | TC-H 106 | BRD-4657

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Pimelic Diphenylamide 106 (orb1223589)

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200 mg
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5 mg
$ 90.00
10 mg
$ 120.00
25 mg
$ 180.00
50 mg
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100 mg
$ 490.00