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Icenticaftor

SKU: orb1298063

Description

Icenticaftor

Research Area

Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number1334546-77-8
MW361.24
Purity98.39%
FormulaC12H13F6N3O3
SMILESCOc1nc(C(=O)NC[C@](C)(O)C(F)(F)F)c(N)cc1C(F)(F)F
TargetCFTR
SolubilityDMSO:150 mg/mL (415.24 mM)

Bioactivity

Target IC50
F508del CFTR:79 nM(EC50)|CFTR (G551D):497 nM(EC50)

Storage & Handling

StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

Alternative Names

QBW 251, QBW251, QBW-251, inhibit, oral, Inhibitor, Icenticaftor, F508del, F508del-CFTR, fibrosis, G551D, G551D-CFTR, CFTR, COPD, cystic, Cystic fibrosis transmembrane conductance regulator

Similar Products

  • Icenticaftor [orb1940188]

    >98% (HPLC)

    1334546-77-8

    361.244

    C12H13F6N3O3

    1 g, 500 mg, 200 mg, 50 mg, 100 mg, 5 mg, 10 mg, 25 mg
Quality Guarantee

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Key Properties

No computed properties available.

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Icenticaftor (orb1298063)

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% DMSO +
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%

Available Sizes

Select a size below

1 mg
$ 210.00
1 ml x 10 mM (in DMSO)
$ 320.00
5 mg
$ 390.00
10 mg
$ 570.00
25 mg
$ 880.00
50 mg
$ 1,210.00
100 mg
$ 1,700.00
200 mg
$ 2,290.00
DispatchUsually dispatched within 3-5 working days
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