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ERα degrader 8

SKU: orb2564543

Description

ERα degrader8 (Compound 18j) is a selective estrogen receptor alpha (ERα) degrading agent. It demonstrates potent anti-proliferative activity in MCF-7 breast cancer cells with an IC50 of 0.15 µM, supporting its use in vitro for cancer research and the study of targeted protein degradation.

Research Area

Metabolism Research

Images & Validation

Key Properties

CAS Number2971837-95-1
MW439.46
FormulaC27H21NO5
SMILESO(C=1C2=C(N=CC1C(=O)C3=C(CC)C=CC=C3)C=C(O)C=C2)C4=CC=C(/C=C/C(O)=O)C=C4
TargetEstrogen Receptor/ERR

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Quality Guarantee

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Key Properties

No computed properties available.

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ERα degrader 8 (orb2564543)

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