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EGFR kinase inhibitor 5

SKU: orb3134123

Description

EGFRkinase inhibitor 5 (Compound 4c) is an orally active epidermal growth factor receptor (EGFR) kinase inhibitor with an IC50 of 18.35 μM. It induces apoptosis and exhibits anticancer and anti-inflammatory properties while maintaining low toxicity (LD50 range of 500-2000 mg/kg).

Research Area

Pharmacology & Drug Discovery; Cell Biology

Images & Validation

Key Properties

FormulaC21H16BrN3OS2
TargetEGFR,Apoptosis

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Protocol Information

EGFR kinase inhibitor 5 (orb3134123)

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