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CPI-0610
Catalog Number: orb1089389
| Catalog Number | orb1089389 |
|---|---|
| Category | Small Molecules |
| Description | CPI-0610 is a small molecule inhibitor of the Bromodomain and Extra-Terminal (BET) family of proteins, with potential antineoplastic activity. Upon administration, the BET inhibitor CPI-0610 binds to the acetylated lysine recognition motifs on the bromodomain of BET proteins, thereby preventing the interaction between the BET proteins and acetylated histone peptides. This disrupts chromatin remodeling and gene expression. Prevention of the expression of certain growth-promoting genes may lead to an inhibition of tumor cell growth. |
| MW | 365.812943458557 |
| CAS Number | [1380087-89-7] |
| Formula | C20H16CLN3O2 |
| SMILES | ClC1=CC=C(C2=N[C@@]([H])(CC(O)=N)C3ON=C(C)C=3C3=CC=CC=C23)C=C1 |
| Note | For research use only |
CPI-0610 carboxylic acid [orb1709989]
98.62%
1380089-81-5
366.8
C20H15ClN2O3
100 mg, 50 mg, 5 mg, 1 mg, 10 mg, 25 mg
