CPI-0610 carboxylic acid

SKU: orb1709989

Description

CPI-0610 carboxylic acid is a potent and selective BET bromodomain inhibitor, serving as a ligand for PROTAC development. It exhibits anticancer activity in preclinical studies, demonstrating efficacy in both in vitro cellular assays and in vivo tumor models.

Research Area

Epigenetics & Chromatin, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 1380089-81-5
• MW: 366.8
• Purity: 98.62%
• Formula: C₂₀H₁₅ClN₂O₃
• SMILES: CC=1C=2C=3C(C(=N[C@@H](CC(O)=O)C2ON1)C4=CC=C(Cl)C=C4)=CC=CC3
• Target: Epigenetic Reader Domain,Ligands for Target Protein for PROTAC

Storage & Handling

• Storage: Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

LigandsforTargetProteinforPROTAC, Ligands for Target Protein for PROTAC, EpigeneticReaderDomain, Epigenetic Reader Domain, CPI0610 carboxylic acid, CPI-0610 carboxylic acid, CPI 0610 carboxylic acid, BET

Compound Identifiers

PubChem CID

67815062