BMS986187

SKU: orb1298464

Description

BMS986187 is a potent and selective positive allosteric modulator (PAM) of the delta-opioid receptor (δ-OR). It is a valuable research tool for investigating δ-OR pharmacology in both in vitro assays and in vivo models of pain, mood, and addiction.

Research Area

Metabolism Research, Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 684238-37-7
• MW: 470.6
• Purity: 99.19%
• Formula: C₃₁H₃₄O₄
• SMILES: Cc1ccccc1COc1ccc(cc1)C1C2=C(CC(C)(C)CC2=O)OC2=C1C(=O)CC(C)(C)C2
• Target: Opioid Receptor
• Solubility: DMSO:4.72 mg/mL (10.03 mM)

Storage & Handling

• Storage: Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

CHO-OPRD1 cell, BMS986187, BMS-986187, BMS 986187, leu-enkephalin, Inhibitor, endomorphin 1, OpioidReceptor, Opioid Receptor, PAM, inhibit, μ-receptor, δ-opioid, δ-opioid receptor

Compound Identifiers

PubChem CID

17379334