VPC-13789

SKU: orb1688383

Description

VPC-13789 is a potent, selective, and orally bioavailable antiandrogen, demonstrating promise for castration-resistant prostate cancer (CRPC) research. It inhibits androgen receptor transcriptional activity in LNCaP cells with an IC50 of 0.19 µM. Its profile supports investigation in both in vitro mechanistic studies and in vivo xenograft models for therapeutic development.

Research Area

Metabolism Research

Key Properties

• CAS Number: 2761146-51-2
• MW: 383.37
• Formula: C₂₁H₁₆F₃N₃O
• SMILES: FC1=C2C(C(=CN2)C3=NC4=C(C=C3)C(C(NC(C)C)=O)=CC=C4)=CC(F)=C1F
• Target: Androgen Receptor,Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

163321994