UFP-803

SKU: orb1679249

Description

This compound is a urotensin-II receptor ligand that acts primarily as a silent antagonist, displaying competitive antagonism in rat aorta (pIC50 = 7.46) and inhibiting U-II-induced plasma extravasation in mice. It is a valuable research tool for investigating the UT receptor system in cardiovascular and renal pathophysiology, both in vitro and in vivo.

Research Area

Metabolism Research, Pharmacology & Drug Discovery

Key Properties

• Target: GPCR
• CAS Number: 879497-82-2
• MW: 1061.24
• Formula: C₅₀H₆₄N₁₀O₁₂S₂
• SMILES: C(C=1C=2C(NC1)=CC=CC2)[C@H]3NC(=O)[C@H](CC4=CC=CC=C4)NC(=O)[C@@H](NC([C@H](CC(O)=O)N)=O)C(C)(C)SSC[C@@H](C(N[C@@H](C(C)C)C(O)=O)=O)NC(=O)[C@H](CC5=CC=C(O)C=C5)NC(=O)[C@H](CCN)NC3=O

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

56972202