UFP-101

SKU: orb1679248

Description

This compound is a potent, selective, and competitive silent antagonist of the NOP receptor, exhibiting high affinity (pKi = 10.24) and over 3000-fold selectivity against classical opioid receptors. It is a valuable research tool for investigating nociceptin's role in pain, anxiety, and addiction pathways, demonstrating antinociceptive effects and blocking nociceptin action in vivo.

Research Area

Metabolism Research, Neuroscience, Pharmacology & Drug Discovery

Key Properties

• Target: Opioid Receptor
• CAS Number: 849024-68-6
• MW: 1908.19
• Formula: C₈₂H₁₃₈N₃₂O₂₁
• SMILES: [C@H](CC1=CC=CC=C1)(C(N[C@H](C(NCC(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@@H](CCC(N)=O)C(N)=O)=O)CC(N)=O)=O)CCCCN)=O)CCCNC(=N)N)=O)CCCCN)=O)CCCNC(=N)N)=O)C)=O)CO)=O)CCCCN)=O)CCCNC(=N)N)=O)C)=O)=O)[C@@H](C)O)=O)NC(CNC(CNC(CNCC2=CC=CC=C2)=O)=O)=O

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

16152632