U-93631

SKU: orb1226154

Description

A potent GABAA receptor antagonist that binds the picrotoxin site and stabilizes the inactive form of the channel via allosteric interaction; induce a rapid, time-dependent decay of GABA-induced whole-cell Cl- currents in recombinant GABAA receptors.

Key Properties

• CAS Number: 152273-12-6
• MW: 299.3676
• Purity: >98% (HPLC)
• Formula: C₁₇H₂₁N₃O₂
• SMILES: O=C(C1=C2N(C=N1)C3=C(C=CC=C3)NC2(C)C)OC(C)(C)C
• Target: GAT
• Solubility: DMSO: ≥ 34 mg/mL

Storage & Handling

• Storage: Storage temperature: -20°C. Stability: ≥ 2 years
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

U93631 | U 93631

Quick Database Links

Gene Symbol

GAT