TRV120056 acetate

SKU: orb1303234

Description

TRV120056 acetate is a Gq-biased angiotensin II type 1 receptor (AT1R) agonist, demonstrating approximately 10-fold greater potency in Gq-mediated signaling compared to β-arrestin-2 pathways. This selective profile makes it a valuable research tool for investigating biased agonism, Gq-dependent physiological and pathological processes in cardiovascular research, both in cellular and animal models.

Key Properties

• Target: Others
• Molecular Weight: 1016.11
• Purity: 99.16%
• Formula: C₄₅H₆₉N₁₃O₁₄
• SMILES: O=C(N(CCC1)[C@@H]1C(NCC(O)=O)=O)[C@@H](NC([C@@]([C@H](C)CC)([H])NC([C@@H](NC([C@@H](C(C)C)NC([C@@H](CCCNC(N)=N)NC([C@@H](N)CC(O)=O)=O)=O)=O)CC2=CC=C(O)C=C2)=O)=O)CC3=CNC=N3.CC(O)=O

Storage & Handling

• Storage: keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

40678-47-5, 40678-47-5 Free base, TRV 120056 Acetate, TRV120056 acetate, TRV120056 Acetate, TRV-120056 Acetate, TRV120056 acetate (40678-47-5 Free base)

Compound Identifiers

PubChem CID

168013235