Tedatioxetine hydrobromide

SKU: orb1708394

Description

Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a multi-target agent functioning as a triple monoamine reuptake inhibitor and a receptor antagonist at several serotonin and adrenergic sites. Its pharmacological profile supports its investigation in preclinical research for depression and anxiety disorders, utilizing both in vitro binding assays and in vivo behavioral models.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 960151-65-9
• MW: 364.34
• Purity: 99.65% (May vary between batches)
• Formula: C₁₈H₂₂BrNS
• SMILES: Br.Cc1ccc(Sc2ccccc2C2CCNCC2)cc1
• Target: Dopamine Receptor,Norepinephrine,Adrenergic Receptor,5-HT Receptor
• Solubility: DMSO:80 mg/mL (219.58 mM);10% DMSO+40% PEG300+5% Tween 80+45% Saline:3.3 mg/mL (9.06 mM)

Bioactivity

• In Vitro:
  Tedatioxetine hydrobromide is often used as an antagonist of 5-HT2A, 5-HT2C, 5-HT3, and α1A adrenergic receptors.

Storage & Handling

• Storage: keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

Dopamine, Dopamine Receptor, DopamineReceptor, 5-HT2A Receptor, 5HT Receptor, 5-HT, 5HTReceptor, Norepinephrine (NE), Lu AA 24530 hydrobromide, Lu AA24530 Hydrobromide, Lu AA-24530 Hydrobromide

Compound Identifiers

PubChem CID

24751582