TD-0212

SKU: orb1708383

Description

TD-0212 is an orally bioavailable small molecule that functions as a dual-acting antagonist of the angiotensin II type 1 receptor (AT1) and an inhibitor of neprilysin (NEP), with respective pKi and pIC50 values of 8.9 and 9.2. This dual pharmacology makes it a valuable research tool for investigating cardiovascular and renal pathophysiology in both in vitro and in vivo experimental models.

Research Area

Metabolism Research

Key Properties

• CAS Number: 1073549-10-6
• MW: 527.65
• Formula: C₂₈H₃₄FN₃O₄S
• SMILES: C(N1C(CNC([C@H](CC(C)C)S)=O)=C(CC)N=C1OCC)C2=C(F)C=C(C=C2)C3=C(C(O)=O)C=CC=C3
• Target: RAAS,Others,Neprilysin

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

45102601