TC14012 TFA

• Catalog Number: orb1981650
• Category: Small Molecules
• Description: TC14012 TFA, a serum-stable derivative of T140, is a selective peptidomimetic CXCR4 antagonist with an IC50 value of 19.3 nM and also functions as a potent CXCR7 agonist, exhibiting an EC50 of 350 nM for recruiting β-arrestin 2 to CXCR7. This compound demonstrates anti-HIV and anti-cancer activities [1] [2].
• Purity: 98.00%
• MW: 2180.44
• Biological Activity: TC14012 TFA, a serum-stable derivative of T140, is a selective peptidomimetic CXCR4 antagonist with an IC50 value of 19.3 nM. It also acts as a potent CXCR7 agonist, exhibiting an EC50 of 350 nM for recruiting β-arrestin 2 to CXCR7. This compound demonstrates anti-HIV and anti-cancer activities [1] [2].
• Formula: C₉₂H₁₄₁F₃N₃₄O₂₁S₂
• Storage: -20°C
• Note: For research use only