Tazemetostat de(methyl morpholine)-COOH

SKU: orb2279009

Description

Tazemetostat de(methyl morpholine)-COOH (compound 7) is a versatile EZH2-directed ligand for constructing PROTAC degraders. These degraders demonstrate potent anti-proliferative activity in both in vitro and in vivo models of diffuse large B-cell lymphoma and other lymphomas, making them valuable research tools for targeted protein degradation studies.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 2685873-44-1
• MW: 517.62
• Formula: C₃₀H₃₅N₃O₅
• SMILES: O=C(O)C=1C=CC(=CC1)C2=CC(C(=O)NCC=3C(=O)NC(=CC3C)C)=C(C(=C2)N(CC)C4CCOCC4)C
• Target: Ligands for Target Protein for PROTAC

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

165437231