(S,R,S)-AHPC-PEG3-N3

SKU: orb1307444

Description

(S,R,S)-AHPC-PEG3-N3

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 1797406-80-4
• MW: 645.77
• Purity: 98.47%
• Formula: C₃₀H₄₃N₇O₇S
• SMILES: C([C@@H](NC(COCCOCCOCCN=[N+]=[N-])=O)[C@](C)(C)C)(=O)N1[C@H](C(NCC2=CC=C(C=C2)C=3SC=NC3C)=O)C[C@@H](O)C1
• Target: E3 Ligase Ligand-Linker Conjugate,Ligand for E3 Ligase
• Solubility: DMSO:50 mg/mL (77.43 mM)

Bioactivity

• In Vitro:
  (S,R,S)-AHPC-PEG3-N3 is derived from patent WO/2016/146985A1, figure 11. PROTAC features an A-L-B structure that tethers a bromodomain inhibitor, binding a BET family protein, to a s All molecule E3 ubiquitin ligase protein binding li and via a suitable linke [1.

Storage & Handling

• Storage: store at low temperature | Pure form: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Disclaimer: For research use only

Alternative Names

VH032-PEG3-N3, VHL, VHL Ligand-Linker Conjugates 8, (S,R,S) AHPC PEG3 N3, (S,R,S)AHPCPEG3N3, (S,R,S)-AHPC-PEG-3-N3, AHPC-PEG3-N3, E3LigaseLigandLinkerConjugate, E3 Ligase Ligand-Linker Conjugate, E3 Ligase Ligand-Linker Conjugates, E3 Ligase LigandLinker Conjugate, E3 ligase Ligand-Linker Conjugates 12, Ligand for E3 Ligase, LigandforE3Ligase, inhibit, Inhibitor

Compound Identifiers

PubChem CID

122539916