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Sodium Channel inhibitor 1

SKU: orb1708501

Description

Sodium Channel inhibitor1 is a novel, selective voltage-gated sodium channel blocker targeting Na v1.7, with IC50 values of 0.16 µM and 0.41 µM at a V hold of -90 mV. It serves as a valuable research tool for investigating pain pathways in both in vitro electrophysiology studies and in vivo preclinical models of nociception.

Research Area

Pharmacology & Drug Discovery

Images & Validation

Key Properties

CAS Number1198117-23-5
MW473.42
FormulaC24H19F4N3O3
SMILESFc1cccc2C(=O)N(CCc3ccccn3)C(C(=O)NCc3ccc(OC(F)(F)F)cc3)c12
TargetSodium Channel,Others

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only

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Key Properties

No computed properties available.

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Sodium Channel inhibitor 1 (orb1708501)

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