SNT-207858

SKU: orb1708503

Description

SNT-207858 is a potent, orally bioavailable, and brain-penetrant selective antagonist of the melanocortin-4 receptor (MC4R), exhibiting IC₅₀ values of 22 nM in binding and 11 nM in functional assays. This compound is a valuable research tool for investigating energy homeostasis and obesity in both in vitro and in vivo models.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 1104080-42-3
• MW: 689.54
• Formula: C₃₂H₄₅Cl₄N₅O₃
• SMILES: CC[C@@H](N1CCCC1)COC2=C(C3CCN(CC3)C([C@H](NC(N4CCCC4)=O)CC5=C(C=C(C=C5)Cl)Cl)=O)N=CC=C2.Cl.Cl
• Target: Melanocortin Receptor,Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

42630199