Saclofen

• Catalog Number: orb1302858
• Category: Small Molecules
• Description: Saclofen
• CAS Number: 125464-42-8
• Purity: 99.54%
• MW: 249.71
• SMILES: C(CS(=O)(=O)O)(CN)C1=CC=C(Cl)C=C1
• Formula: C₉H₁₂ClNO₃S
• Biological Activity: Saclofen is a sulfonic analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA) that acts as a competitive antagonist of the GABAB receptor (IC50: 7.8 μM).1 This compound can be used to determine the functional roles for the GABAB receptor as a mediator of slow inhibitory postsynaptic potentials in the brain.
• Note: For research use only
• Expiration Date: 12 months from date of receipt.