Pinacidil monohydrate

SKU: orb1219640

Description

Pinacidil monohydrate is a potassium channel activator, antihypertensive drug.Pinacidil hydrate activates the ATP-modulated potassium channels of guinea pog bladder and heart with Ki of 104 and 251 nM, respectively.(In Vitro):Pinacidil monohydrate is a potassium channel activator. Pinacidil hydrate is an antihypertensive drug of the class of agents called "potassium channel openers". Pinacidil hydrate activates the ATP-modulated potassium channels of guinea pog bladder and heart with Ki values of 104 and 251 nM, respectively.

Key Properties

• CAS Number: 85371-64-8
• MW: 263.34
• Purity: >98% (HPLC)
• Formula: C₁₃H₂₁N₅O
• SMILES: O.CC(N\C(NC#N)=N\c1ccncc1)C(C)(C)C
• Target: Potassium Channel
• Solubility: DMSO:97 mg/mL (368.35mM; Need ultrasonic); Ethanol:47 mg/mL (178.48mM; Need ultrasonic)

Bioactivity

• In Vitro:
  Pinacidil monohydrate is a potassium channel activator. Pinacidil hydrate is an antihypertensive drug of the class of agents called "potassium channel openers". Pinacidil hydrate activates the ATP-modulated potassium channels of guinea pog bladder and heart with Ki values of 104 and 251 nM, respectively.

Storage & Handling

• Storage: Storage temperature: -20°C. Stability: ≥ 2 years
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Quick Database Links

Gene Symbol

Potassium Channel