L-R4W2

SKU: orb1679417

Description

This potent and selective TRPV1 antagonist peptide exhibits an IC50 of approximately 0.1 µM, effectively inhibiting calcium influx in dorsal root ganglion neurons in vitro. It serves as a valuable research tool for studying pain pathways and has demonstrated analgesic efficacy in animal models.

Research Area

Pharmacology & Drug Discovery

Key Properties

• Target: TRP/TRPV Channel
• CAS Number: 206350-79-0
• MW: 1014.2
• Formula: C₄₆H₇₁N₂₁O₆
• SMILES: C([C@@H](C(N[C@@H](CC=1C=2C(NC1)=CC=CC2)C(N)=O)=O)NC([C@@H](NC([C@@H](NC([C@@H](NC([C@H](CCCNC(=N)N)N)=O)CCCNC(=N)N)=O)CCCNC(=N)N)=O)CCCNC(=N)N)=O)C=3C=4C(NC3)=CC=CC4

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

90479804