Kisspeptin 234

SKU: orb1679451

Description

Kisspeptin 234 is a synthetic kisspeptin-10 analog that acts as a potent antagonist of the kisspeptin receptor (KISS1R/GPR54). It inhibits kisspeptin-stimulated inositol phosphate production (IC50 = 7 nM) and GnRH release. This tool compound is widely used in vitro and in vivo to study the neuroendocrine regulation of reproduction.

Research Area

Pharmacology & Drug Discovery

Key Properties

• Target: Kisspeptin
• CAS Number: 1145998-81-7
• MW: 1295.42
• Formula: C₆₃H₇₈N₁₈O₁₃
• SMILES: C([C@H](NC([C@@H](NC([C@H](NC(C)=O)C)=O)CC(N)=O)=O)C(N[C@H](C(NCC(N[C@@H](CC1=CC=CC=C1)C(NCC(N[C@H](CC=2C=3C(NC2)=CC=CC3)C(N[C@H](C(N[C@@H](CC4=CC=CC=C4)C(N)=O)=O)CCCNC(=N)N)=O)=O)=O)=O)=O)CC(N)=O)=O)C=5C=6C(NC5)=CC=CC6

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

90488890