ERAP2-IN-1

SKU: orb1687182

Description

ERAP2-IN-1 (compound 61) is a selective, non-competitive inhibitor of the aminopeptidase ERAP2, blocking its activity against fluorogenic and peptide substrates with IC50 values of 27 μM and 44 μM, respectively. This tool compound is useful for studying ERAP2's role in antigen processing, both in biochemical and cellular assays.

Research Area

Metabolism Research

Key Properties

• CAS Number: 2420551-38-6
• MW: 458.45
• Formula: C₂₀H₂₁F₃N₂O₅S
• SMILES: N(S(=O)(=O)C1=C(OC)C=CC(C(O)=O)=C1)C2=C(C=C(C(F)(F)F)C=C2)N3CCCCC3
• Target: Aminopeptidase,Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

85470736