ERAP1-IN-1

SKU: orb1309692

Description

ERAP1-IN-1

Research Area

Metabolism Research

Key Properties

• CAS Number: 865273-97-8
• MW: 458.45
• Purity: 98.60%
• Formula: C₂₀H₂₁F₃N₂O₅S
• SMILES: COc1ccc(cc1S(=O)(=O)Nc1cc(ccc1N1CCCCC1)C(F)(F)F)C(O)=O
• Target: Aminopeptidase,Others
• Solubility: 10% DMSO+90% Corn Oil:3.3 mg/mL (7.2 mM);DMSO:250 mg/mL (545.32 mM)

Bioactivity

• In Vitro:
  ERAP1-IN-1 (50 μM) exhibits specific inhibition of ERAP1 in the cellular context. ERAP1-IN-1 allosterically activates ERAP1’s hydrolysis of fluorogenic and chromogenic amino acid substrates.

Storage & Handling

• Storage: Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

inhibit, Inhibitor, ERAP1 IN 1, ERAP1IN1, ERAP-1-IN-1, ERAP1-IN-1, ERAP1, endoplasmic, aminopeptidase, reticulum

Compound Identifiers

PubChem CID

4798291