Elinogrel

SKU: orb1309711

Description

Elinogrel (PRT060128) is a potent, competitive, and reversible P2Y12 receptor antagonist with an IC50 of 20 nM. It is a valuable research tool for studying antiplatelet mechanisms and has demonstrated efficacy in preclinical models of thrombosis, supporting both in vitro and in vivo cardiovascular research.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 936500-94-6
• MW: 523.95
• Purity: 97.09% (May vary between batches)
• Formula: C₂₀H₁₅ClFN₅O₅S₂
• SMILES: CNc1cc2[nH]c(=O)n(-c3ccc(NC(=O)NS(=O)(=O)c4ccc(Cl)s4)cc3)c(=O)c2cc1F
• Target: P2Y Receptor
• Solubility: 10% DMSO+40% PEG300+5% Tween 80+45% Saline:4 mg/mL (7.63 mM);DMSO:120 mg/mL (229.03 mM)

Bioactivity

• Target IC50:
  P2Y12:20 nM

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

Inhibitor, Elinogrel, inhibit, PRT 060128, PRT060128, PRT-060128, P2YReceptor, P2Y Receptor, P2Y12

Compound Identifiers

PubChem CID

16066663