ELA-11(human)

SKU: orb1679428

Description

This high-affinity apelin receptor agonist (Ki=14 nM) is a bioactive ELA-32 fragment that inhibits forskolin-induced cAMP production and stimulates β-arrestin recruitment in vitro. It is utilized in research on apelin signaling, including cardiovascular and metabolic disease studies.

Research Area

Cardiovascular Research, Pharmacology & Drug Discovery

Key Properties

• Target: Arrestin,Apelin receptor
• CAS Number: 1784687-32-6
• MW: 1283.57
• Formula: C₅₈H₉₀N₁₆O₁₃S₂
• SMILES: C(N[C@H](C(=O)N1[C@H](C(O)=O)CCC1)CC2=CC=CC=C2)(=O)[C@H]3N(C([C@@H](NC([C@@H](NC([C@@H](NC([C@H](CC4=CN=CN4)NC([C@@H](NC(=O)[C@H]5N(C([C@@H](NC([C@H](CS)N)=O)CCSC)=O)CCC5)CC(C)C)=O)=O)CO)=O)CCCNC(=N)N)=O)[C@@H](C)C)=O)CCC3

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

127043376