d[Leu4,Lys8]-VP

SKU: orb1679424

Description

This compound is a selective vasopressin V1B receptor agonist with Ki values of 0.16 nM for V1B, 64 nM for OT, 100 nM for V2, and 3800 nM for V1A receptors. It exhibits minimal antidiuretic, vasopressor, and oxytocic activity, making it a valuable research tool for studying V1B receptor function in stress, anxiety, and depression models both in vitro and in vivo.

Research Area

Pharmacology & Drug Discovery

Key Properties

• Target: Vasopressin Receptor
• CAS Number: 42061-33-6
• MW: 1026.2
• Formula: C₄₇H₆₇N₁₁O₁₁S₂
• SMILES: C(=O)(N1[C@H](C(N[C@H](C(NCC(N)=O)=O)CCCCN)=O)CCC1)[C@H]2NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC3=CC=CC=C3)NC(=O)[C@H](CC4=CC=C(O)C=C4)NC(=O)CCSSC2

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

44419030