(D-Arg8)-Inotocin

SKU: orb2277343

Description

(D-Arg⁸)-Inotocin is a highly potent and selective competitive antagonist of the vasopressin V1a receptor, with a Ki of 1.3 nM and >3000-fold selectivity over related receptors. It is a valuable research tool for investigating the physiological and pathological roles of V1aR signaling in both in vitro binding assays and in vivo animal studies.

Research Area

Pharmacology & Drug Discovery

Key Properties

• Target: Vasopressin Receptor
• CAS Number: 745816-74-4
• MW: 973.17
• Formula: C₃₉H₆₈N₁₄O₁₁S₂
• SMILES: C(=O)(N1[C@H](C(N[C@@H](C(NCC(N)=O)=O)CCCNC(=N)N)=O)CCC1)[C@H]2NC(=O)[C@H](CC(N)=O)NC(=O)[C@]([C@@H](C)O)(NC(=O)[C@]([C@H](CC)C)(NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)CSSC2)[H])[H]

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

168432158