CTAP

SKU: orb2692712

Description

CTAP is a potent, highly selective, and BBB penetrant μ opioid receptor antagonist, with an IC50 of 3.5 nM. CTAP displays over 1200-fold selectivity over δ opioid (IC50=4500 nM) and somatostatin receptors. CTAP can be used for the study of L-DOPA-induced dyskinesia (LID) and opiate overdose or addiction.

Key Properties

• Target: Opioid Receptor
• CAS Number: 103429-32-9
• MW: 1102.33
• Purity: ≥95%
• Formula: C₅₁H₆₇N₁₃O₁₁S
• Protein Sequence: {D-Phe}-CY-{D-Trp}-RT-{Pen}-T-NH2 (Disulfide bridge:Cys2-Pen7)

Storage & Handling

• Expiration Date: 6 months from date of receipt.
• Disclaimer: For research use only

Quick Database Links

Gene Symbol

Opioid Receptor