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CS-VIP 8 TFA

SKU: orb3027791

Description

CS-VIP 8 TFA is a selective allosteric inhibitor of the WDR5 protein (Ki= 0.008 μM). It induces a conformational change in the MLL1 complex, leading to the dissociation of MLL1 from the complex, thereby inhibiting the MLL1 histone methyltransferase activity and modulating HOX gene expression. CS-VIP 8 TFA shows potential for research in hematological disorders such as leukemia.

Research Area

Immunology & Inflammation

Images & Validation

Key Properties

FormulaC45H53F7N12O9
TargetJAK,Histone Methyltransferase

Storage & Handling

Storage-20°C
Expiration Date12 months from date of receipt.
DisclaimerFor research use only
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Protocol Information

CS-VIP 8 TFA (orb3027791)

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