BQ-3020 ammonium

• Catalog Number: orb2278874
• Category: Small Molecules
• Description: BQ-3020 ammonium, a selective endothelin receptor (ET B receptor) agonist, demonstrates inhibition of [125 I] ET-1 binding to ET B receptors with an IC50 of 0.2 nM and induces vasoconstriction in rabbit pulmonary arteries. Additionally, it promotes relaxation of the pig urinary bladder neck, rendering it useful for research into cardiovascular diseases [1] [2].
• Purity: 98.00%
• MW: 2006.32 (free base)
• Biological Activity: BQ-3020 ammonium, a selective endothelin receptor (ET B receptor) agonist, demonstrates inhibition of [125 I] ET-1 binding to ET B receptors with an IC50 of 0.2 nM and induces vasoconstriction in rabbit pulmonary arteries. Additionally, it promotes relaxation of the pig urinary bladder neck, rendering it useful for research into cardiovascular diseases [1] [2].
• Formula: C₉₆H₁₄₀N₂₀O₂₅S.xNH₃
• Storage: -20°C
• Note: For research use only