Azaperol-D4

SKU: orb2655269

Description

Azaperone-d4 is the deuterium labeled Azaperone. Azaperone (R-1929) acts as a dopamine antagonist but also has some antihistaminic and anticholinergic properties. Azaperone is a pyridinylpiperazine and butyrophenone neuroleptic agent with antiemetic effects, which is used mainly as a tranquilizer in veterinary medicine.Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs.

Key Properties

• CAS Number: 1173021-72-1
• MW: 331.42
• Purity: >98% (HPLC)
• Formula: C₁₉H₁₈D₄FN₃O
• SMILES: O=C(C1=C([2H])C([2H])=C(C([2H])=C1[2H])F)CCCN2CCN(C3=CC=CC=N3)CC2

Bioactivity

• In Vitro:
  Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs.

Storage & Handling

• Storage: Storage temperature: -20°C. Stability: ≥ 2 years
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

R-1929-d4