Apelin-17(human, bovine)

SKU: orb1679260

Description

This small molecule is a potent endogenous agonist of the apelin receptor, demonstrating high activity with a pIC50 of 9.94 in inhibiting forskolin-induced cAMP production in vitro. It is a valuable research tool for studying cardiovascular function, metabolism, and fluid homeostasis in both cellular and animal models.

Research Area

Infectious Disease & Virology, Pharmacology & Drug Discovery, Protein Biochemistry

Key Properties

• Target: Apelin receptor,HIV Protease
• CAS Number: 217082-57-0
• MW: 2138.56
• Formula: C₉₆H₁₅₆N₃₄O₂₀S
• SMILES: C([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@H](CC1=CC=CC=C1)NC([C@H](CCCCN)N)=O)=O)CCCNC(=N)N)=O)CCCNC(=N)N)=O)CCC(N)=O)=O)CCCNC(=N)N)(=O)N2[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@@H](CC3=CN=CN3)C(N[C@H](C(NCC(=O)N4[C@H](C(N[C@H](C(=O)N5[C@H](C(N[C@@H](CC6=CC=CC=C6)C(O)=O)=O)CCC5)CCSC)=O)CCC4)=O)CCCCN)=O)=O)CO)=O)CC(C)C)=O)CCCNC(=N)N)=O)CCC2

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

16130452