A 841720

• Catalog Number: orb1704946
• Category: Small Molecules
• Description: A 841720
• CAS Number: 869802-58-4
• Purity: 98%
• MW: 343.45
• SMILES: N(C)(C)C1=C2C3=C(SC2=NC=C1)C(=O)N(C=N3)N4CCCCCC4
• Formula: C₁₇H₂₁N₅OS
• Biological Activity: A-841720 is a potent, selective, and non-competitive antagonist of the mGlu1 receptor, exhibiting an IC 50 value of 10 nM specifically for the human mGlu1 receptor. It demonstrates a 34-fold greater selectivity for mGlu1 over mGlu5 (IC 50 of 342 nM), with negligible activity across a spectrum of other neurotransmitter receptors, ion channels, and transporters. Additionally, A-841720 possesses analgesic potential within a certain dose range [1] [2].
• Note: For research use only
• Expiration Date: 12 months from date of receipt.