ELA-11 (human) acetate(1784687-32-6 free base)

SKU: orb1296435

Description

ELA-11 (human) acetate is a bioactive apelin receptor fragment derived from ELA-32, acting as a high-affinity agonist (Ki = 14 nM). It demonstrates functional activity by inhibiting forskolin-stimulated cAMP production and promoting β-arrestin recruitment in vitro, making it a valuable tool for studying APJ receptor signaling in cardiovascular and metabolic research.

Research Area

Pharmacology & Drug Discovery

Key Properties

• Target: Apelin receptor,Arrestin
• Molecular Weight: 1343.61
• Purity: 99.53%
• Formula: C₆₀H₉₄N₁₆O₁₅S₂
• SMILES: O=C(N1[C@@H](CCC1)C(O)=O)[C@H](CC2=CC=CC=C2)NC([C@H]3N(CCC3)C([C@H](C(C)C)NC([C@H](CCCNC(N)=N)NC([C@H](CO)NC([C@@H](NC([C@H](CC(C)C)NC([C@H]4N(CCC4)C([C@H](CCSC)NC([C@@H](N)CS)=O)=O)=O)=O)CC5=CN=CN5)=O)=O)=O)=O)=O.CC(O)=O

Storage & Handling

• Storage: keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Alternative Names

Apelinreceptor, Apelin receptor, ELA-11 acetate(1784687-32-6 free base), ELA11 (human) acetate(1784687326 free base), ELA 11 (human) acetate(1784687 32 6 free base)

Compound Identifiers

PubChem CID

169553468