APJ receptor agonist 6

SKU: orb1686369

Description

APJ receptor agonist 6 is a potent small molecule agonist for the apelin receptor, demonstrating high binding affinity (Ki: 0.059 µM) and functional activity (EC50: 6.22 µM). This compound is a valuable research tool for investigating APJ receptor signaling in cardiovascular and metabolic disease models, both in vitro and in vivo.

Research Area

Cardiovascular Research; Pharmacology & Drug Discovery, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 1965244-85-2
• MW: 523.6
• Formula: C₂₉H₃₄FN₃O₅
• SMILES: O(C)C1=C(C=2N(N=C(C(N[C@@H](CCC3CCCCC3)CC(O)=O)=O)C2)C4=CC=C(F)C=C4)C(OC)=CC=C1
• Target: Apelin receptor,Others,Arrestin

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

127051280