RXFP1 receptor agonist-4

SKU: orb1943521

Description

RXFP1 receptor agonist-4 (Example 268) is a potent small molecule agonist of the human RXFP1 receptor, exhibiting an EC50 of 4.9 nM for cAMP suppression in stable HEK293 cell assays. This compound is a valuable research tool for investigating relaxin receptor signaling in both cellular and animal models of fibrosis and cardiovascular disease.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 2941376-76-5
• MW: 695.6
• Formula: C₃₂H₂₄F₇N₃O₅S
• SMILES: O=C(NC1=CC=C(F)C(=C1)C(F)(F)F)C=2SC=3C=C(C=CC3C2NC(=O)C=4C=C(C=CC4OC)C5=NOC6CC(CO)CC56)C(F)(F)F
• Target: RXFP receptor,Others

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

168476180