L-803087

SKU: orb1785931

Description

L-803087 is a potent and selective somatostatin sst4 receptor agonist with a Ki of 0.7 nM, which is > 280-fold higher than other somatostatin receptors. L-803087 facilitates AMPA-mediated hippocampal synaptic responses in vitro and increases kainate-induced seizures in mice.

Key Properties

• CAS Number: 217480-26-7
• MW: 599.55
• Purity: >98%
• Formula: C₂₅H₂₉F₂N₅O₃
• SMILES: NC(NCCCC(C(OC)=O)NC(CCCC1=C(C2=CC=CC=C2)NC2=C(C=C(C=C12)F)F)=O)=N.OC(C(F)(F)F)=O

Storage & Handling

• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only