DA-302168S

SKU: orb3028215

Description

DA-302168S is an orally active, selective GLP-1R agonist with an EC50 value of 1.32 nM. It promotes insulin secretion and has a hypoglycemic effect. Additionally, DA-302168S reduces food intake. It primarily activates GLP-1R in humans and monkeys, with minimal effect on GLP-1R in rats, mice, and dogs. DA-302168S can be used for research in type 2 diabetes and obesity.

Research Area

Pharmacology & Drug Discovery

Key Properties

• CAS Number: 2969158-02-7
• MW: 616.011
• Formula: C₃₃H₂₄ClF₂N₃O₅
• SMILES: C(N1C=2C(N=C1CC3=C(F)C=C(C=C3)C=4N=C(OCC5=C6C(C=CO6)=C(Cl)C=C5)C(F)=CC4)=CC=C(C(O)=O)C2)[C@@H]7CCO7
• Target: Glucagon Receptor

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Quick Database Links

Gene Symbol

Glucagon Receptor