Lys-[Des-Arg9]Bradykinin

SKU: orb1679432

Description

This endogenous peptide is a potent and highly selective bradykinin B1 receptor agonist, exhibiting a Ki of 0.12 nM at the human B1 receptor versus >30,000 nM at B2. It acts as a hypotensive agent by reducing peripheral vascular resistance in vivo and is a valuable research tool for studying inflammation, pain, and cardiovascular pharmacology in both in vitro and in vivo models.

Research Area

Musculoskeletal & Connective Tissue Research, Pharmacology & Drug Discovery

Key Properties

• Target: Bradykinin Receptor
• CAS Number: 71800-36-7
• MW: 1032.21
• Formula: C₅₀H₇₃N₁₃O₁₁
• SMILES: C(=O)([C@H]1N(C([C@@H](NC([C@H](CCCCN)N)=O)CCCNC(=N)N)=O)CCC1)N2[C@H](C(NCC(N[C@@H](CC3=CC=CC=C3)C(N[C@H](C(=O)N4[C@H](C(N[C@@H](CC5=CC=CC=C5)C(O)=O)=O)CCC4)CO)=O)=O)=O)CCC2

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

122227