Cart summary

You have no items in your shopping cart.

    PF-04979064

    PF-04979064

    Catalog Number: orb341528

    DispatchUsually dispatched within 5-10 working days
    $ 1,377.00
    Catalog Numberorb341528
    CategorySmall Molecules
    DescriptionPF-04979064 is a highly potent and orally bioavailable PI3K/mTOR dual inhibitor developed through structure-based drug design. It inhibited mTOR, PI3Kα, β, δ and γ isoforms and AKT phosphorylation with IC50 as 2.64 nM, 0.395 nM, 0.111 nM, 0.122 nM and 28.
    CAS Number[1220699-06-8]
    MW446.5
    SMILESC[C@@H](C(N1CCC(N2C(=O)N(C)C3=CN=C4C=CC(C5C=CC(C)=NC=5)=NC4=C23)CC1)=O)O
    FormulaC24H26N6O3
    NoteFor research use only
    Expiration Date12 months from date of receipt.
    • PF-04979064 [orb1226766]

      > 98% (HPLC)

      1220699-06-8

      100 mg, 50 mg, 25 mg, 10 mg, 5 mg, 2 mg, 1 g, 500 mg, 200 mg
    • PF-04979064 [orb1299901]

      98%

      1220699-06-8

      446.5

      C24H26N6O3

      10 mg, 25 mg, 50 mg, 5 mg, 2 mg
    • PF-04979064 [orb1897922]

      1220699-06-8

      5 mg
    • PF-04979064 [orb1897923]

      1220699-06-8

      2 mg
    • PF-04979064 [orb1897924]

      1220699-06-8

      10 mg
    Submit a review

    Filter by Rating

      • Star
      • Star
      • Star
      • Star
      • Star
      • 5 stars
      • Star
      • Star
      • Star
      • Star
      • Star
      • 4 stars
      • Star
      • Star
      • Star
      • Star
      • Star
      • 3 stars
      • Star
      • Star
      • Star
      • Star
      • Star
      • 2 stars
      • Star
      • Star
      • Star
      • Star
      • Star
      • 1 stars