K-(D-1-Nal)-FwLL-NH2 TFA

SKU: orb1981509

Description

K-(D-1-Nal)-FwLL-NH₂ TFA is a high-affinity inverse agonist of the ghrelin receptor (GHSR1a), with Ki values of 4.9 nM and 31 nM in cellular assays. It potently inhibits Gq and G13 signaling pathways, making it a valuable tool for in vitro and in vivo research into metabolic disorders and appetite regulation.

Research Area

Immunology & Inflammation; Metabolism Research, Pharmacology & Drug Discovery

Key Properties

• Target: GHSR
• MW: 1016.16
• Formula: C₅₃H₆₈F₃N₉O₈

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Quick Database Links

Gene Symbol

GHSR