ZINC02092166

• Catalog Number: orb1473025
• Category: Small Molecules
• Description: ZINC02092166 is a novel potent, and selective small-molecule inhibitor for the β-catenin/Tcf4 protein-protein interaction with Ki of 1.7 and 7.0 uM in AlphaScreen and FP assay (wild-type β-catenin), respectively; remain affinity for muant catenin V511S, V511S/I569S and R469A with Ki of 20-50 uM; exhibits dual selectivity for β-catenin/Tcf over β-catenin/cadherin and β-catenin/APC PPIs.
• CAS Number: [354543-09-2]
• MW: 349.26388001442
• SMILES: O1N=C2C(N1)=NC1=C(C3C=CC=CC=3C1=N2)/N=N/C(C1C(N)=NON=1)=O
• Formula: C₁₄H₇N₉O₃
• Note: For research use only
• Expiration Date: 12 months from date of receipt.