SR48692

• Catalog Number: orb146169
• Category: Small Molecules
• Description: SR 48692 is a neurotensin antagonist; selective for NTS1 over NTS2 (apparent affinity, Ke, is 36 nM for NTS1). Competitively inhibits binding of [125I]-neurotensin to HT29 and N1E115 cell membranes (IC50 values are 15.3 and 20.4 nM respectively).
• CAS Number: [146362-70-1]
• MW: 587.06534
• SMILES: COC1=C(C(OC)=CC=C1)C2N(N=C(C=2)C(=O)NC3(C(O)=O)C4CC5CC3CC(C5)C4)C6C7C(=CC(Cl)=CC=7)N=CC=6
• Formula: C₃₂H₃₁N₄O₅CL
• Note: For research use only
• Expiration Date: 12 months from date of receipt.