SB 242084 dihydrochloride

SKU: orb1693152

Description

SB 242084 hydrochloride is a potent and selective 5-HT2C receptor antagonist with a pKi of 9.0, exhibiting 158-fold and 100-fold selectivity over 5-HT2A and 5-HT2B receptors, respectively. This compound is a valuable pharmacological tool used in vitro and in vivo to investigate the role of 5-HT2C receptors in anxiety, depression, and feeding behavior.

Research Area

Neuroscience, Pharmacology & Drug Discovery

Key Properties

• CAS Number: 1049747-87-6
• MW: 467.78
• Purity: 97.01% (May vary between batches)
• Formula: C₂₁H₂₁Cl₃N₄O₂
• SMILES: O=C(N1C2=CC(Cl)=C(C)C=C2CC1)NC3=CN=C(C=C3)OC4=CC=CN=C4C.Cl.Cl
• Target: 5-HT Receptor

Storage & Handling

• Storage: -20°C
• Expiration Date: 12 months from date of receipt.
• Disclaimer: For research use only

Compound Identifiers

PubChem CID

16219981